唐薰,李筱芳,王家坡,杨新国
湖南省科技计划项目资助课题! ( 962 -4 3 )
TANG Xun,LI Xiao fang,WANG Jia po,YANG Xing guo
以N-苯基-2,6-二氯苯胺为起始原料,经酰胺化,环合,水解开环得目标产物,总收率达74%。工艺简单,产品质量好,可较大幅度降低成本。
The new process,from the starting material N phenyl 2,6 dichloroaniline through chloroacetylation,cyclization and hydrolysis,gained 73 % total yield.It is comparably simple,with better quality of the product and much lower costs.
唐薰,李筱芳,王家坡,杨新国.制备双氯灭痛的新工艺研究[J].湖南大学学报:自然科学版,2000,27(3):